Abstract
A series of tetrahydroisoquinolines has yielded potent MT(2) receptor antagonists, which are selective versus the MT(1) receptor.
MeSH terms
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Humans
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Protein Binding / physiology
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Receptor, Melatonin, MT2 / antagonists & inhibitors*
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Receptor, Melatonin, MT2 / metabolism*
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Tetrahydroisoquinolines / chemistry*
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Tetrahydroisoquinolines / metabolism*
Substances
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Receptor, Melatonin, MT2
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Tetrahydroisoquinolines